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Found 289 Enz. Inhib. hit(s) with Target = 'Regulator of G-protein signaling 8'
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM46590(4-[2-[(E)-(2,3-dihydroxy-4-oxocyclohexa-2,5-dien-1...)
Affinity DataKi:  20nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM32274(2,5-bis(chloranyl)-3-(4-methylpiperazin-1-yl)-6-(2...)
Affinity DataKi:  20nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM38361(2-(4-pyrrolidin-1-ylsulfonylphenyl)-1,2-benzothiaz...)
Affinity DataKi:  20nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataKi:  60nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM33097(3-[[7-(1,3-benzothiazol-2-ylsulfanyl)-4-nitro-2,1,...)
Affinity DataKi:  70nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM40728(2-[2-oxidanylidene-2-[2-[(Z)-(3-oxidanyl-4-oxidany...)
Affinity DataKi:  100nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47719((4-chlorodithiazol-5-ylidene)-(4-chloro-2-methyl-p...)
Affinity DataKi:  110nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM34435(4-cyano-3-methyl-5-[[1-oxo-2-[[5-(phenylmethyl)-1,...)
Affinity DataKi:  150nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47815(2-(4-Methoxy-phenyl)-[1,4]benzoquinone | 2-(4-meth...)
Affinity DataKi:  150nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47735(3-chloranyl-N-(3,3-dimethylbutan-2-yl)-6-nitro-1-b...)
Affinity DataKi:  170nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM46608((4E)-5-methyl-4-[(3-nitroanilino)methylene]-2-phen...)
Affinity DataKi:  180nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM34702((4E)-2,3-dihydroxy-4-[[(4-methyl-2-methylimino-1,3...)
Affinity DataKi:  260nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM34972(MLS000759648 | N''-[(E)-(2,3-dihydroxy-4-oxo-1-cyc...)
Affinity DataKi:  320nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM33145(3-[[[(E)-(2,3-dihydroxy-4-keto-cyclohexa-2,5-dien-...)
Affinity DataKi:  340nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM62209(UNM-0000305796 | cid_18559023)
Affinity DataKi:  400nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47764((4E)-5-methyl-4-[[3-[[(Z)-(3-methyl-1-phenyl-5-sul...)
Affinity DataKi:  430nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM34524(2-[2-keto-2-[3-methyl-4-(m-tolyl)piperazino]ethyl]...)
Affinity DataKi:  460nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM33090((4E)-4-[[(2-ethylimino-4-methyl-1,3-thiazol-3-yl)a...)
Affinity DataKi:  470nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47776(3-chloranyl-N-(3-morpholin-4-ylpropyl)-6-nitro-1-b...)
Affinity DataKi:  470nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47770(4-[5-[(2,2-dimethyl-4,6-dioxo-1,3-dioxan-5-ylidene...)
Affinity DataKi:  580nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47696(4-[(3-carbamoyl-4,5-dimethyl-2-thienyl)amino]-4-ke...)
Affinity DataKi:  700nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47747(4-[(E)-[3-[3-(diethylsulfamoyl)phenyl]-5-thioxo-1H...)
Affinity DataKi:  2.59E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM62216(2-(4,6-dimethylisothiazolo[5,4-b]pyridin-3-yl)oxy-...)
Affinity DataKi:  2.64E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47734(MLS000553854 | N-[(4-methylphenyl)-(5-nitro-8-oxid...)
Affinity DataKi:  3.59E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384745(CHEMBL2037237)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384744(CHEMBL2037236)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384775(CHEMBL2037227)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384741(CHEMBL2037232)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384743(CHEMBL2037235)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384776(CHEMBL2037228)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384767(CHEMBL2037365)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384761(CHEMBL2037358)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384764(CHEMBL2037362)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384757(CHEMBL2037354)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384750(CHEMBL2037349)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50:  1.10E+4nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384777(CHEMBL2037229)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384755(CHEMBL2037352)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384752(CHEMBL2037351)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384746(CHEMBL2037238)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384742(CHEMBL2037233)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384747(CHEMBL2037346)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384759(CHEMBL2037356)
Affinity DataIC50:  1.57E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384740(CHEMBL2037231)
Affinity DataIC50:  1.62E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384748(CHEMBL2037347)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384778(CHEMBL2037230)
Affinity DataIC50:  1.72E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384756(CHEMBL2037353)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384739(CHEMBL2037357)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50384751(CHEMBL2037350)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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